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atazanavir

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EntityQ423467· pop 28· linked from 153 articles

atazanavir

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Also known as CGP-73547, ATZ, ATV, Zrivada, Latazanavir, Atazanavirum

Atazanavir, sold under the brand name Reyataz among others, is an antiretroviral medication used to treat HIV/AIDS. It is generally recommended for use with other antiretrovirals. It may be used for post-exposure prophylaxis after a needlestick injury or other potential exposure. It is taken by mouth.

Chemical data

Formula
C38H52N6O7
Molecular weight
704.9 g/mol
IUPAC name
methyl N-[(2S)-1-[2-[(2S,3S)-2-hydroxy-3-[[(2S)-2-(methoxycarbonylamino)-3,3-dimethylbutanoyl]amino]-4-phenylbutyl]-2-[(4-pyridin-2-ylphenyl)methyl]hydrazinyl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate
SMILES
CC(C)(C)[C@@H](C(=O)N[C@@H](CC1=CC=CC=C1)[C@H](CN(CC2=CC=C(C=C2)C3=CC=CC=N3)NC(=O)[C@H](C(C)(C)C)NC(=O)OC)O)NC(=O)OC
InChIKey
AXRYRYVKAWYZBR-GASGPIRDSA-N
XLogP
5.6
Polar surface area
171 Ų
H-bond donors
5
H-bond acceptors
9
Formal charge
0

via PubChem

~7 min read

Encyclopedic overview

7 sections
Contents
  • Medical uses
  • Pregnancy
  • Contraindications
  • Adverse effects
  • Mechanism of action
  • Synthesis
  • References

{{Drugbox | Verifiedfields = changed | verifiedrevid = 458476502 | image = Atazanavir structure.svg | image_class = skin-invert-image | width = 180 | alt = | image2 = Atazanavir ball-and-stick.png | image_class2 = bg-transparent | width2 = 220 | alt2 =

| pronounce = | tradename = Reyataz, Evotaz, others | Drugs.com = | MedlinePlus = a603019 | DailyMedID = Atazanavir | pregnancy_AU = B2 | pregnancy_AU_comment = | routes_of_administration = By mouth | ATC_prefix = J05 | ATC_suffix = AE08 | ATC_supplemental =

Excerpted from Wikipedia’s “atazanavir” article, available under the CC BY-SA 4.0 licence.

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