ensaculin
Sign in to saveEnsaculin (KA-672) is a drug from the coumarin family, which has been researched as a potential treatment for dementia. It acts on a number of receptor systems, being both a weak NMDA antagonist and a 5HT1A agonist. Animal studies have shown promising nootropic effects, although efficacy in humans has yet to be proven. It was well tolerated in human trials, with the main side effect being orthostatic hypotension (low blood pressure upon standing).
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 452.231
Show 3 more facts
- chemical formula
- C₂₆H₃₂N₂O₅
- canonical SMILES
- CC1=C(C(=O)OC2=CC(=C(C=C12)OCCCN3CCN(CC3)C4=CC=CC=C4OC)OC)C
- subject has role
- nootropic
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Ensaculin (KA-672) is a drug from the coumarin family, which has been researched as a potential treatment for dementia. It acts on a number of receptor systems, being both a weak NMDA antagonist and a 5HT1A agonist. Animal studies have shown promising nootropic effects, although efficacy in humans has yet to be proven. It was well tolerated in human trials, with the main side effect being orthostatic hypotension (low blood pressure upon standing).
==See also== Enciprazine Mafoprazine BMY-14802 Azaperone Fluanisone
Excerpted from Wikipedia’s “ensaculin” article, available under the CC BY-SA 4.0 licence.