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valproic acid

File:2-propylpentanoic_acid_200.svg · Wikimedia Commons · See Wikimedia Commons

EntityQ240642· pop 43· linked from 1,979 articles

valproic acid

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Also known as LEP321, A-44090, 2-n-propyl-n-valeric acid, n-DPA, DPA, dipropylacetic acid, VPA, 2-n-propyl-4-pentenoic acid

Valproate (valproic acid, VPA, sodium valproate, and valproate semisodium forms) are medications primarily used to treat epilepsy and as a mood stabilizer in the treatment of bipolar disorder. They are useful for the prevention of seizures in those with absence seizures, partial seizures, and generalized seizures. They can be given intravenously or by mouth, and the tablet forms exist in both long- and short-acting formulations.

OverviewAI-generated

Valproic acid, also identified as 2-propylpentanoic acid, is a chemical compound with the formula C₈H₁₆O₂. It has a mass of 144.115 and a density of 0.904. The substance melts at 25 degrees and boils at 221.5 degrees. Its inception is recorded as 1967.

Chemical properties include a charge of 0, an xlogp of 2.8, and a tpsa of 37.3. The molecule contains one hydrogen bond donor and two hydrogen bond acceptors. PubChem lists its weight as 144.21.

The compound is referenced by 1,979 other encyclopedia articles. A PubMed query for valproic acid yields a count of 19638.

Synthesized by Vinony from 22 facts across 4 sources: Wikidata, PubMed, PubChem, Vinony graph. Generated from structured data (not the Wikipedia text) and checked against those facts — may still contain errors.

Key facts

Drug.metabolism
Liver—glucuronide conjugation 30–50%, mitochondrial β-oxidation over 40%
Drug.elimination_half life
9–16 hours
Drug.excretion
Urine (30–50%)
Drug.CAS_number
76584-70-8
Drug.PubChem
23663956
Drug.IUPHAR_ligand
7009
Drug.DrugBank
DBSALT000185
Drug.ChemSpiderID
48337
Drug.UNII
644VL95AO6
Drug.KEGG
D00304
Drug.ChEBI
4667
Drug.ChEMBL
2105613
Drug.Watchedfields
changed
Drug.verifiedrevid
464404696
Drug.image
Sodium-valproate-2D-skeletal.png
Drug.image_class
skin-invert-image
Drug.width
250
Drug.image2
Valproato Sódico.png

via Wikipedia infobox

Chemical data

Formula
C8H16O2
Molecular weight
144.21 g/mol
IUPAC name
2-propylpentanoic acid
SMILES
CCCC(CCC)C(=O)O
InChIKey
NIJJYAXOARWZEE-UHFFFAOYSA-N
XLogP
2.8
Polar surface area
37.3 Ų
H-bond donors
1
H-bond acceptors
2
Formal charge
0

via PubChem

Research

19,638 papers

via PubMed

Wikidata facts

Mass
144.115
Show 10 more facts
found in taxon
Valeriana officinalis
chemical formula
C₈H₁₆O₂
World Health Organisation international non-proprietary name
valproic acid
canonical SMILES
CCCC(CCC)C(=O)O
Commons category
Valproic acid
legal status (medicine)
boxed warning
inception
1967-00-00
melting point
25
boiling point
221.5
density
0.904
Sources (9)

via Wikidata · CC0

~29 min read

Encyclopedic overview

45 sections
Contents
  • Medical uses
  • Epilepsy
  • Psychiatric disorders
  • Other uses
  • Contraindications
  • Adverse effects
  • Pregnancy
  • Elderly
  • Overdose and toxicity
  • Interactions
  • Pharmacology
  • Pharmacodynamics
  • Endocrine actions
  • Pharmacokinetics
  • Chemistry
  • History
  • Society and culture
  • Restrictions
  • Approval status
  • Off-label uses
  • Formulations
  • Terminology
  • Brand names of valproic acid
  • Brand names of sodium valproate
  • Portugal
  • United States
  • Australia
  • New Zealand
  • UK
  • UK only
  • Germany, Switzerland, Norway, Finland, Sweden
  • South Africa
  • Malaysia
  • Romania
  • Canada
  • Japan
  • Europe
  • Taiwan
  • Iran
  • Israel
  • India, Russia and [[Commonwealth of Independent States|CIS]] countries
  • Uruguay
  • Brand names of valproate semisodium
  • Research
  • References

Valproate (valproic acid, VPA, sodium valproate, and valproate semisodium forms) are medications primarily used to treat epilepsy and as a mood stabilizer in the treatment of bipolar disorder. They are useful for the prevention of seizures in those with absence seizures, partial seizures, and generalized seizures. They can be given intravenously or by mouth, and the tablet forms exist in both long- and short-acting formulations.

Common side effects of valproate include nausea, vomiting, somnolence, and dry mouth. Serious side effects can include liver failure, and regular monitoring of liver function tests is therefore recommended. Other serious risks include pancreatitis and an increased suicide risk.

Excerpted from Wikipedia’s “valproic acid” article, available under the CC BY-SA 4.0 licence.

Gallery (16)