berotralstat

Also known as Orladeyo, BCX7353

Berotralstat, sold under the brand name Orladeyo, is a medication used to prevent attacks of hereditary angioedema. Berotralstat is a plasma kallikrein inhibitor. It is taken by mouth.

Key facts

Drug.image: Berotralstat Structure.svg
Drug.image_class: skin-invert-image
Drug.tradename: Orladeyo
Drug.DailyMedID: Berotralstat
Drug.routes_of_administration: By mouth
Drug.class: Plasma kallikrein inhibitor
Drug.ATC_prefix: B06
Drug.ATC_suffix: AC06
Drug.legal_CA: Rx-only
Drug.legal_US: Rx-only
Drug.legal_EU: Rx-only
Drug.index2_label: as HCl
Drug.CAS_number: 1809010-50-1
Drug.CAS_number2: 1809010-52-3
Drug.PubChem: 137528262
Drug.DrugBank: DB15982
Drug.ChemSpiderID: 81368516
Drug.UNII: XZA0KB1BDQ

via Wikipedia infobox

Wikidata facts

Mass: 562.210422332

Show 3 more facts

canonical SMILES: C1CC1CNC(C2=CC(=C(C=C2)F)NC(=O)C3=CC(=NN3C4=CC=CC(=C4)CN)C(F)(F)F)C5=CC=CC(=C5)C#N
isomeric SMILES: C1CC1CN[C@@H](C2=CC(=C(C=C2)F)NC(=O)C3=CC(=NN3C4=CC=CC(=C4)CN)C(F)(F)F)C5=CC=CC(=C5)C#N
chemical formula: C₃₀H₂₆F₄N₆O

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Article

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Contents

Medical uses
History
Society and culture
Legal status
Names
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Berotralstat, sold under the brand name Orladeyo, is a medication used to prevent attacks of hereditary angioedema. Berotralstat is a plasma kallikrein inhibitor. It is taken by mouth.

The most common side effects include abdominal pain, vomiting, diarrhea, back pain, and heartburn.