etizolam
Sign in to savethumb|Etizolam powder. Pictured is roughly 150 mg; a standard dose is around 1 mg alt=Four blister packs of Etizex brand etizolam tablets|thumb|Etizex brand etizolam tablets Etizolam is a thienodiazepine derivative which is a benzodiazepine analog. The etizolam molecule differs from a benzodiazepine in that the benzene ring has been replaced by a thiophene ring and triazole ring has been fused, making the drug a thienotriazolodiazepine.
Key facts
- Drug.Verifiedfields
- changed
- Drug.Watchedfields
- changed
- Drug.verifiedrevid
- 443854261
- Drug.IUPAC_name
- 4-(2-Chlorophenyl)-2-ethyl-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine
- Drug.tradename
- Etizest, Etilaam, Etizex, Depas, Sedekopan, Pasaden
- Drug.image
- Etizolam.svg
- Drug.image_class
- skin-invert-image
- Drug.width
- 150
- Drug.image2
- Etizolam-from-xtal-3D-bs-17.png
- Drug.image_class2
- bg-transparent
- Drug.KEGG
- D01514
- Drug.ChemSpiderID
- 3191
- Drug.smiles
- ClC1=CC=CC=C1C2=NCC3=NN=C(C)N3C4=C2C=C(CC)S4
- Drug.StdInChI
- 1S/C17H15ClN4S/c1-3-11-8-13-16(12-6-4-5-7-14(12)18)19-9-15-21-20-10(2)22(15)17(13)23-11/h4-8H,3,9H2,1-2H3
- Drug.StdInChIKey
- VMZUTJCNQWMAGF-UHFFFAOYSA-N
- Drug.UNII
- A76XI0HL37
- Drug.CAS_number
- 40054-69-1
- Drug.ATC_prefix
- N05
via Wikipedia infobox
Research
259 papers- Etizolam.2006
- Etizolam: A rapid review on pharmacology, non-medical use and harms.Drug and alcohol review · 2020
- Etizolam and Its Major Metabolites: A Short Review.Journal of analytical toxicology · 2023
- "Pressed" Etizolam.The Journal of pediatrics · 2021
- Etizolam and Irish drug poisoning deaths.Irish journal of psychological medicine · 2024
via PubMed
Article
20 sectionsContents
- Medical uses
- Side effects
- Tolerance, dependence and withdrawal
- Pharmacology
- Interactions
- Overdose
- Society and culture
- Brand names
- Legal status
- International drug control conventions
- Australia
- Denmark
- Germany
- Italy
- India
- United States
- Misuse
- See also
- References
- External links
thumb|Etizolam powder. Pictured is roughly 150 mg; a standard dose is around 1 mg alt=Four blister packs of Etizex brand etizolam tablets|thumb|Etizex brand etizolam tablets Etizolam is a thienodiazepine derivative which is a benzodiazepine analog. The etizolam molecule differs from a benzodiazepine in that the benzene ring has been replaced by a thiophene ring and triazole ring has been fused, making the drug a thienotriazolodiazepine.
Although a thienodiazepine, etizolam is clinically regarded as a benzodiazepine because of its mode of action via the benzodiazepine receptor and directly targeting GABAA allosteric modulator receptors.
Gallery (3)
Connections
Categories
2-Chlorophenyl compoundsChemical pages without DrugBank identifierDesigner drugsDrugboxes which contain changes to verified fieldsDrugboxes which contain changes to watched fieldsECHA InfoCard ID from WikidataGABAA receptor positive allosteric modulatorsHallucinogen antidotesHypnoticsInfobox drug articles with non-default infobox titleThienotriazolodiazepines