ezlopitant
Sign in to saveAlso known as CJ 11974, CJ-11974, CJ11974
Ezlopitant (INN, code name CJ-11,974) is an NK1 receptor antagonist. It has antiemetic and antinociceptive effects. Pfizer was developing ezlopitant for the treatment of irritable bowel syndrome but it appears to have been discontinued.
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 454.298414
Show 4 more facts
- chemical formula
- C₃₁H₃₈N₂O
- isomeric SMILES
- CC(C)C1=CC(=C(C=C1)OC)CN[C@@H]2[C@@H](N3CCC2CC3)C(C4=CC=CC=C4)C5=CC=CC=C5
- canonical SMILES
- CC(C)C1=CC(=C(C=C1)OC)CNC2C3CCN(C2C(C4=CC=CC=C4)C5=CC=CC=C5)CC3
- Commons category
- Ezlopitant
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Encyclopedic overview
2 sectionsContents
- See also
- References
Ezlopitant (INN, code name CJ-11,974) is an NK1 receptor antagonist. It has antiemetic and antinociceptive effects. Pfizer was developing ezlopitant for the treatment of irritable bowel syndrome but it appears to have been discontinued.
== See also == NK1 receptor antagonist Maropitant (tert-butyl instead of isopropyl)
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