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natalizumab
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natalizumab

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Also known as AN100226m, PB006, anti-alpha4 integrin, anti-VLA4, antegran, natalizumab-sztn

Natalizumab, sold under the brand name Tysabri among others, is a medication used to treat multiple sclerosis and Crohn's disease. It is a humanized monoclonal antibody against the cell adhesion molecule α4-integrin. It is given by intravenous infusion. The drug is believed to work by reducing the ability of inflammatory immune cells to attach to and pass through the cell layers lining the intestines and blood–brain barrier.

Key facts

Drug.Verifiedfields
changed
Drug.Watchedfields
changed
Drug.verifiedrevid
458283255
Drug.type
mab
Drug.image
Natalizumab 4IRZ.png
Drug.caption
Natalizumab Fab fragment bound to the headpiece of an α4-integrin. From PDB .
Drug.mab_type
mab
Drug.source
zu/o
Drug.target
alpha-4 integrin
Drug.tradename
Tysabri, others
Drug.MedlinePlus
a605006
Drug.DailyMedID
Natalizumab
Drug.pregnancy_AU
C
Drug.routes_of_administration
Intravenous
Drug.ATC_prefix
L04
Drug.ATC_suffix
AG03
Drug.biosimilars
natalizumab-sztn, Tyruko
Drug.legal_AU
S4

via Wikipedia infobox

Research

3,689 papers

via PubMed

Wikidata facts

Subclass of
protein
Has use
medication
Show 8 more facts
route of administration
intravenous infusion and defusion
World Health Organisation international non-proprietary name
natalizumab
defined daily dose
10
subject has role
monoclonal antibody
medical condition treated
Crohn's disease
has characteristic
biopharmaceutical
legal status (medicine)
boxed warning
side effect
nausea
Sources (5)

via Wikidata · CC0

~14 min read

Encyclopedic overview

12 sections
Contents
  • Medical uses
  • Adverse effects
  • Mechanism of action
  • Multiple sclerosis
  • Crohn's disease
  • Interactions
  • History
  • Society and culture
  • Legal status
  • Biosimilars
  • References
  • Further reading

Natalizumab, sold under the brand name Tysabri among others, is a medication used to treat multiple sclerosis and Crohn's disease. It is a humanized monoclonal antibody against the cell adhesion molecule α4-integrin. It is given by intravenous infusion. The drug is believed to work by reducing the ability of inflammatory immune cells to attach to and pass through the cell layers lining the intestines and blood–brain barrier.

Natalizumab is a monoclonal antibody which targets a protein called α4β1 integrin on white blood cells involved in inflammation. By attaching to integrin, natalizumab is thought to stop white blood cells from entering the brain and spinal cord tissue, thereby reducing inflammation and the resulting nerve damage.

Excerpted from Wikipedia’s “natalizumab” article, available under the CC BY-SA 4.0 licence.

Gallery (2)