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zenazocine
Sign in to saveZenazocine (INN; WIN-42,964) is an opioid analgesic of the benzomorphan family which made it to phase II clinical trials before development was ultimately halted and it was never marketed. It acts as a partial agonist of the μ- and δ-opioid receptors, with less intrinsic activity at the former receptor and more at the latter receptor (hence, it behaves more antagonistically at the former and more agonistically at the latter), and produces antinociceptive effects in animal studies.
In the Vinony graph
Within Vinony's link graph, zenazocine is referenced by 694 other articles, and connects out to (+)-catechin, butorphanol and International Standard Book Number.
It is catalogued under topics including Benzomorphans, Chemical pages without DrugBank identifier and Drugs not assigned an ATC code.
Its subject is documented across 4 Wikipedia language editions.
Chemical data
- Formula
- C23H35NO2
- Molecular weight
- 357.5 g/mol
- IUPAC name
- 1-[(1S,9R)-4-hydroxy-1,10,13-trimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-13-yl]-6-methylheptan-3-one
- SMILES
- CC(C)CCC(=O)CCC1([C@H]2CC3=C([C@@]1(CCN2C)C)C=C(C=C3)O)C
- InChIKey
- JZFZEWWOIOYBTQ-AXWGZAFASA-N
- XLogP
- 4.7
- Polar surface area
- 40.5 Ų
- H-bond donors
- 1
- H-bond acceptors
- 3
- Formal charge
- 0
via PubChem
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 357.266779
Show 4 more facts
- chemical formula
- C₂₃H₃₅NO₂
- canonical SMILES
- CC(C)CCC(=O)CCC1(C2CC3=C(C1(CCN2C)C)C=C(C=C3)O)C
- isomeric SMILES
- CC(C)CCC(=O)CCC1([C@H]2CC3=C([C@@]1(CCN2C)C)C=C(C=C3)O)C
- Commons category
- Zenazocine
Sources (1)
via Wikidata · CC0
~1 min read
Encyclopedic overview
2 sectionsContents
- See also
- References
Zenazocine (INN; WIN-42,964) is an opioid analgesic of the benzomorphan family which made it to phase II clinical trials before development was ultimately halted and it was never marketed. It acts as a partial agonist of the μ- and δ-opioid receptors, with less intrinsic activity at the former receptor and more at the latter receptor (hence, it behaves more antagonistically at the former and more agonistically at the latter), and produces antinociceptive effects in animal studies.
== See also == Tonazocine
Excerpted from Wikipedia’s “zenazocine” article, available under the CC BY-SA 4.0 licence.