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carbimazole

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Also known as Athyromazole, Ethyl 3-methyl-2-thioimidazoline-1-carboxylate, Carbethoxymethimazole, Carbimazolo, Carbinazole, Thyrostat, Carbimazol, Carbimazolum

Carbimazole (brand names Neo-Mercazole, Anti-Thyrox, etc.) is used to treat hyperthyroidism. Carbimazole is a pro-drug as after absorption it is converted to the active form, methimazole. Methimazole prevents thyroid peroxidase enzyme from iodinating and coupling the tyrosine residues on thyroglobulin, hence reducing the production of the thyroid hormones T3 and T4 (thyroxine).

Research

1,666 papers

via PubMed

~3 min read

Encyclopedic overview

6 sections
Contents
  • Medical uses
  • Adverse effects
  • Precautions
  • Brand names
  • References
  • Further reading

Carbimazole (brand names Neo-Mercazole, Anti-Thyrox, etc.) is used to treat hyperthyroidism. Carbimazole is a pro-drug as after absorption it is converted to the active form, methimazole. Methimazole prevents thyroid peroxidase enzyme from iodinating and coupling the tyrosine residues on thyroglobulin, hence reducing the production of the thyroid hormones T3 and T4 (thyroxine).

It is on the World Health Organization's List of Essential Medicines.

Excerpted from Wikipedia’s “carbimazole” article, available under the CC BY-SA 4.0 licence.