phaclofen
Sign in to savePhaclofen, or phosphonobaclofen, is a selective antagonist for the GABAB receptor. It was the first selective GABAB antagonist discovered, but its utility was limited by the fact that it does not cross the blood brain barrier.
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 249.032158
Show 2 more facts
- chemical formula
- C₉H₁₃ClNO₃P
- canonical SMILES
- C1=CC(=CC=C1C(CN)CP(=O)(O)O)Cl
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Encyclopedic overview
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- References
Phaclofen, or phosphonobaclofen, is a selective antagonist for the GABAB receptor. It was the first selective GABAB antagonist discovered, but its utility was limited by the fact that it does not cross the blood brain barrier.
==References==
Excerpted from Wikipedia’s “phaclofen” article, available under the CC BY-SA 4.0 licence.