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rapacuronium bromide

Structure via PubChem · Public domain (PubChem)

EntityQ3419354· pop 6· linked from 344 articles

rapacuronium bromide

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Also known as ORG-9487, Raplon

pharmaceutical drug

Chemical data

Formula
C37H61BrN2O4
Molecular weight
677.8 g/mol
IUPAC name
[(2S,3S,5S,8R,9S,10S,13S,14S,16S,17R)-3-acetyloxy-10,13-dimethyl-2-piperidin-1-yl-16-(1-prop-2-enylpiperidin-1-ium-1-yl)-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl] propanoate bromide
SMILES
CCC(=O)O[C@H]1[C@H](C[C@@H]2[C@@]1(CC[C@H]3[C@H]2CC[C@@H]4[C@@]3(C[C@@H]([C@H](C4)OC(=O)C)N5CCCCC5)C)C)[N+]6(CCCCC6)CC=C.[Br-]
InChIKey
LVQTUXZKLGXYIU-GWSNJHLMSA-M
Polar surface area
55.8 Ų
H-bond donors
0
H-bond acceptors
6
Formal charge
0

via PubChem

Drug data · ChEMBL

Withdrawn
Max clinical phase
Approved
Molecule type
Small molecule
First approval
1999
Admin. routes
parenteral

via ChEMBL · EBI

Wikidata facts

Has part
bromine
Mass
676.381
Has use
medication
Show 3 more facts
chemical formula
C₃₇H₆₁BrN₂O₄
canonical SMILES
CCC(=O)OC1C(CC2C1(CCC3C2CCC4C3(CC(C(C4)OC(=O)C)N5CCCCC5)C)C)[N+]6(CCCCC6)CC=C.[Br-]
isomeric SMILES
CCC(=O)O[C@H]1[C@H](C[C@@H]2[C@@]1(CC[C@H]3[C@H]2CC[C@@H]4[C@@]3(C[C@@H]([C@H](C4)OC(=O)C)N5CCCCC5)C)C)[N+]6(CCCCC6)CC=C.[Br-]
Sources (2)

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via Wikidata sitelinks · CC0