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EntityQ519447· pop 15· linked from 40 articles

Also known as FX-1006, 2-(3,5-dichlorophenyl)benzoxazole-6-carboxylic acid, tafamidisum

Tafamidis, sold under the brand names Vyndaqel and Vyndamax, is a medication used to delay disease progression in adults with certain forms of transthyretin amyloidosis. It can be used to treat both hereditary forms, familial amyloid cardiomyopathy and familial amyloid polyneuropathy, as well as wild-type transthyretin amyloidosis, which formerly was called senile systemic amyloidosis. It works by stabilizing the quaternary structure of the protein transthyretin. In people with transthyretin amyloidosis, transthyretin falls apart and forms clumps called (amyloid) that harm tissues including ne

Key facts

Drug.Verifiedfields
changed
Drug.Watchedfields
changed
Drug.verifiedrevid
458948015
Drug.image
Tafamidis.svg
Drug.image_class
skin-invert-image
Drug.width
200
Drug.tradename
Vyndaqel, Vyndamax, others
Drug.DailyMedID
Tafamidis
Drug.pregnancy_AU
D
Drug.routes_of_administration
By mouth
Drug.ATC_prefix
N07
Drug.ATC_suffix
XX08
Drug.legal_AU
S4
Drug.legal_CA
Rx-only
Drug.legal_CA_comment
/ Schedule D
Drug.legal_UK
POM
Drug.legal_US
Rx-only
Drug.legal_EU
Rx-only

via Wikipedia infobox

Wikidata facts

Mass
306.98
Show 4 more facts
chemical formula
C₁₄H₇Cl₂NO₃
canonical SMILES
C1=CC2=C(C=C1C(=O)O)OC(=N2)C3=CC(=CC(=C3)Cl)Cl
World Health Organisation international non-proprietary name
tafamidis
defined daily dose
20
Sources (4)

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~6 min read

Article

11 sections
Contents
  • Medical use
  • Adverse effects
  • Interactions
  • Pharmacology
  • Chemistry
  • History
  • Society and culture
  • Legal status
  • Economics
  • References
  • Further reading

Tafamidis, sold under the brand names Vyndaqel and Vyndamax, is a medication used to delay disease progression in adults with certain forms of transthyretin amyloidosis. It can be used to treat both hereditary forms, familial amyloid cardiomyopathy and familial amyloid polyneuropathy, as well as wild-type transthyretin amyloidosis, which formerly was called senile systemic amyloidosis. It works by stabilizing the quaternary structure of the protein transthyretin. In people with transthyretin amyloidosis, transthyretin falls apart and forms clumps called (amyloid) that harm tissues including nerves and the heart.

The US Food and Drug Administration considers tafamidis to be a first-in-class medication.

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