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hydroquinidine

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EntityQ27106893· pop 7· linked from 59 articles

hydroquinidine

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Dihydroquinidine (also called hydroquinidine) is an organic compound, a cinchona alkaloid closely related to quinine. The specific rotation is +226° in ethanol at 2 g/100 ml. A derivative of this molecule is used as chiral ligand in the AD-mix for Sharpless dihydroxylation.

Chemical data

Formula
C20H26N2O2
Molecular weight
326.4 g/mol
IUPAC name
(S)-[(2R,5R)-5-ethyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methoxyquinolin-4-yl)methanol
SMILES
CC[C@H]1CN2CCC1C[C@@H]2[C@H](C3=C4C=C(C=CC4=NC=C3)OC)O
InChIKey
LJOQGZACKSYWCH-NBGVHYBESA-N
XLogP
3.1
Polar surface area
45.6 Ų
H-bond donors
1
H-bond acceptors
4
Formal charge
0

via PubChem

Drug data · ChEMBL

Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
326.199428
Show 4 more facts
canonical SMILES
CCC1CN2CCC1CC2C(C3=C4C=C(C=CC4=NC=C3)OC)O
chemical formula
C₂₀H₂₆N₂O₂
isomeric SMILES
CC[C@H]1CN2CCC1C[C@@H]2[C@H](C3=C4C=C(C=CC4=NC=C3)OC)O
Commons category
Dihydroquinidine
Sources (1)

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Encyclopedic overview

2 sections
Contents
  • See also
  • References

Dihydroquinidine (also called hydroquinidine) is an organic compound, a cinchona alkaloid closely related to quinine. The specific rotation is +226° in ethanol at 2 g/100 ml. A derivative of this molecule is used as chiral ligand in the AD-mix for Sharpless dihydroxylation.

The substance is also a class Ia antiarrhythmic medication.

Excerpted from Wikipedia’s “hydroquinidine” article, available under the CC BY-SA 4.0 licence.

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