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pildralazine

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EntityQ7193849· pop 5· linked from 58 articles

pildralazine

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Also known as propildazine

Pildralazine (Atensil), also known as propyldazine or propildazine, is an antihypertensive and vasodilator.

Chemical data

Formula
C8H15N5O
Molecular weight
197.24 g/mol
IUPAC name
1-[(6-hydrazinylpyridazin-3-yl)-methylamino]propan-2-ol
SMILES
CC(CN(C)C1=NN=C(C=C1)NN)O
InChIKey
KYIAWOXNPBANEW-UHFFFAOYSA-N
XLogP
-0.4
Polar surface area
87.3 Ų
H-bond donors
3
H-bond acceptors
6
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Phase 2
Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
197.128
Show 3 more facts
Commons category
Pildralazine
chemical formula
C₈H₁₅N₅O
canonical SMILES
CC(CN(C)C1=NN=C(C=C1)NN)O
Sources (2)

via Wikidata · CC0

~1 min read

Encyclopedic overview

2 sections
Contents
  • Synthesis
  • References

Pildralazine (Atensil), also known as propyldazine or propildazine, is an antihypertensive and vasodilator.

==Synthesis== [[File:Pildralazine synthesis.svg|thumb|center|500px|class=skin-invert-image|Thieme Synthesis: Patent:]]

Excerpted from Wikipedia’s “pildralazine” article, available under the CC BY-SA 4.0 licence.

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