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minoxidil

File:Minoxidil_structure.svg · Wikimedia Commons · See Wikimedia Commons

EntityQ424165· pop 38· linked from 482 articles

Also known as Rogaine®, 2,4-Diamino-6-piperidinopyrimidine 3-oxide, Minossidile, Minoxidilum, Tricoxidil, Minoximen, Regaine

Minoxidil, sold under the brand names Loniten and Rogaine among others, is a medication used for the treatment of high blood pressure and pattern hair loss. It is an antihypertensive and a vasodilator. It is available as a generic medication by prescription in oral tablet form and over-the-counter as a topical liquid or foam.

Key facts

Drug.image
Minoxidil structure.svg
Drug.image_class
skin-invert-image
Drug.width
150
Drug.alt
A space filling model of the molecule
Drug.image2
Minoxidil-from-xtal-3D-balls.png
Drug.image_class2
bg-transparent
Drug.width2
135
Drug.tradename
Loniten, Rogaine, others
Drug.MedlinePlus
a682608
Drug.DailyMedID
Minoxidil
Drug.pregnancy_AU
C
Drug.routes_of_administration
Oral, sublingual, topical (solution, foam, spray)
Drug.class
Potassium channel opener; KATP channel opener
Drug.ATC_prefix
C02
Drug.ATC_suffix
DC01
Drug.legal_AU
S4
Drug.legal_AU_comment
/ S2
Drug.legal_UK
GSL

via Wikipedia infobox

Chemical data

Formula
C9H15N5O
Molecular weight
209.25 g/mol
IUPAC name
3-hydroxy-2-imino-6-piperidin-1-ylpyrimidin-4-amine
SMILES
C1CCN(CC1)C2=NC(=N)N(C(=C2)N)O
InChIKey
ZIMGGGWCDYVHOY-UHFFFAOYSA-N
XLogP
1.2
Polar surface area
88.9 Ų
H-bond donors
3
H-bond acceptors
3
Formal charge
0

via PubChem

Wikidata facts

Mass
209.1277
Show 6 more facts
chemical formula
C₉H₁₅N₅O
World Health Organisation international non-proprietary name
minoxidil
canonical SMILES
C1=C([N+](=C(N=C1N2CCCCC2)N)[O-])N
defined daily dose
20
MCN code
2933.59.91
Commons category
Minoxidil
Sources (5)

via Wikidata · CC0

~24 min read

Article

31 sections
Contents
  • Medical uses
  • High blood pressure
  • Hair loss
  • Available forms
  • Side effects
  • Overdose
  • Interactions
  • Pharmacology
  • Pharmacodynamics
  • Pharmacokinetics
  • Absorption
  • Distribution
  • Metabolism
  • Elimination
  • Chemistry
  • Properties
  • Synthesis
  • History
  • Initial development
  • Repurposing for hair growth
  • Society and culture
  • Economics
  • Brand names
  • Research
  • Hair loss
  • Beard growth
  • Nail problems
  • Other uses
  • Toxicity to animals
  • References
  • External links

Minoxidil, sold under the brand names Loniten and Rogaine among others, is a medication used for the treatment of high blood pressure and pattern hair loss. It is an antihypertensive and a vasodilator. It is available as a generic medication by prescription in oral tablet form and over-the-counter as a topical liquid or foam.

==Medical uses== ===High blood pressure=== Minoxidil, when used for hypertension, is generally reserved for use in severe hypertension patients who do not respond to at least two agents and a diuretic. Minoxidil is also generally administered with a loop diuretic to prevent sodium retention and potassium retention. It may also cause a reflex tachycardia and thus is prescribed with a beta blocker.

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