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propofol

File:Propofol.svg · Wikimedia Commons · See Wikimedia Commons

EntityQ422740· pop 52· linked from 1,153 articles

Also known as 2,6-diisopropylphenol, ICI 35868, 2,6-bis(1-methylethyl)phenol, 2,6-di(propan-2-yl)phenol

Propofol is the active component of an intravenous anesthetic formulation used for induction and maintenance of general anesthesia. The formulation was approved under the brand name Diprivan. Numerous generic versions have since been released. Intravenous administration is used to induce unconsciousness, after which anesthesia may be maintained using a combination of medications. It is manufactured as part of a sterile injectable emulsion formulation using soybean oil and lecithin, giving it a white milky coloration.

OverviewAI-generated

Propofol is a chemical compound with the formula C₁₂H₁₈O. Its IUPAC name is 2,6-di(propan-2-yl)phenol. The substance has a mass of 178.136 and a density of 0.955. Physical properties include a melting point of 18, a boiling point of 247, and a refractive index of 1.5140.

Chemical analysis indicates that propofol has an xlogp of 3.8 and a tpsa of 20.2. It contains one hydrogen bond donor and one hydrogen bond acceptor, with a charge of 0. The canonical SMILES representation is CC(C)C1=C(C(=CC=C1)C(C)C)O.

The compound is referenced by 1,153 other encyclopedia articles. A search for propofol in PubMed yields a count of 29528.

Synthesized by Vinony from 22 facts across 4 sources: Wikidata, PubMed, PubChem, Vinony graph. Generated from structured data (not the Wikipedia text) and checked against those facts — may still contain errors.

Key facts

Drug.Watchedfields
changed
Drug.verifiedrevid
456484691
Drug.image
Propofol.svg
Drug.image_class
skin-invert-image
Drug.image2
Propofol ball-and-stick model from xtal 2014.png
Drug.image_class2
bg-transparent
Drug.alt2
Ball-and-stick model of propofol
Drug.tradename
Diprivan, others
Drug.DailyMedID
Propofol
Drug.pregnancy_AU
C
Drug.addiction_liability
Moderate
Drug.dependency_liability
Physical: Very high Psychological: no data
Drug.routes_of_administration
Intravenous
Drug.class
GABAA receptor agonist;sedative;general anesthetic
Drug.ATC_prefix
N01
Drug.ATC_suffix
AX10
Drug.legal_AU
S4
Drug.legal_BR
C1

via Wikipedia infobox

Chemical data

Formula
C12H18O
Molecular weight
178.27 g/mol
IUPAC name
2,6-di(propan-2-yl)phenol
SMILES
CC(C)C1=C(C(=CC=C1)C(C)C)O
InChIKey
OLBCVFGFOZPWHH-UHFFFAOYSA-N
XLogP
3.8
Polar surface area
20.2 Ų
H-bond donors
1
H-bond acceptors
1
Formal charge
0

via PubChem

Research

29,528 papers

via PubMed

~17 min read

Encyclopedic overview

21 sections
Contents
  • Uses
  • Anesthesia
  • Routine procedural sedation
  • COVID-19
  • Status epilepticus
  • Other uses
  • Assisted death in Canada
  • Capital punishment
  • Recreational use
  • Manufacturing
  • Side effects
  • Propofol infusion syndrome
  • Interactions
  • Pharmacology
  • Pharmacodynamics
  • Pharmacokinetics
  • History
  • Developments
  • Veterinary uses
  • References
  • External links

Propofol is the active component of an intravenous anesthetic formulation used for induction and maintenance of general anesthesia. The formulation was approved under the brand name Diprivan. Numerous generic versions have since been released. Intravenous administration is used to induce unconsciousness, after which anesthesia may be maintained using a combination of medications. It is manufactured as part of a sterile injectable emulsion formulation using soybean oil and lecithin, giving it a white milky coloration.

Compared to other anesthetic agents, recovery from propofol-induced anesthesia is generally rapid and associated with less frequent side effects (e.g., drowsiness, nausea, vomiting). Propofol may be used prior to diagnostic procedures requiring anesthesia, in the management of refractory status epilepticus, and for induction or maintenance of anesthesia prior to and during surgeries. It may be administered as a bolus or an infusion, or as a combination of the two.

Excerpted from Wikipedia’s “propofol” article, available under the CC BY-SA 4.0 licence.

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