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nerisopam

Structure via PubChem · Public domain (PubChem)

EntityQ6996288· pop 9· linked from 182 articles

Nerisopam (GYKI-52322, EGIS-6775) is a drug which is a 2,3-benzodiazepine derivative, related to tofisopam. It has potent anxiolytic and neuroleptic effects in animal studies.

Chemical data

Formula
C18H19N3O2
Molecular weight
309.4 g/mol
IUPAC name
4-(7,8-dimethoxy-4-methyl-5H-2,3-benzodiazepin-1-yl)aniline
SMILES
CC1=NN=C(C2=CC(=C(C=C2C1)OC)OC)C3=CC=C(C=C3)N
InChIKey
WWQDEXGFYVSTCX-UHFFFAOYSA-N
XLogP
1.6
Polar surface area
69.2 Ų
H-bond donors
1
H-bond acceptors
5
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Phase 2
Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
309.148
Show 3 more facts
chemical formula
C₁₈H₁₉N₃O₂
canonical SMILES
CC1=NN=C(C2=CC(=C(C=C2C1)OC)OC)C3=CC=C(C=C3)N
Commons category
Nerisopam
Sources (2)

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Encyclopedic overview

2 sections
Contents
  • See also
  • References

Nerisopam (GYKI-52322, EGIS-6775) is a drug which is a 2,3-benzodiazepine derivative, related to tofisopam. It has potent anxiolytic and neuroleptic effects in animal studies.

==See also== Benzodiazepine

Excerpted from Wikipedia’s “nerisopam” article, available under the CC BY-SA 4.0 licence.

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