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EntityQ7088466· pop 13· linked from 118 articles

olodaterol

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Also known as BI-1744-CL, Striverdi®, BI 1744, BI-1744

Olodaterol (trade name Striverdi Respimat) is an ultra-long-acting β adrenoreceptor agonist (ultra-LABA) used as an inhalation for treating people with chronic obstructive pulmonary disease (COPD). It is manufactured by Boehringer Ingelheim.

Wikidata facts

Mass
386.184172
Has use
medication
Show 8 more facts
chemical formula
C₂₁H₂₆N₂O₅
canonical SMILES
CC(C)(CC1=CC=C(C=C1)OC)NCC(C2=CC(=CC3=C2OCC(=O)N3)O)O
isomeric SMILES
CC(C)(CC1=CC=C(C=C1)OC)NC[C@@H](C2=CC(=CC3=C2OCC(=O)N3)O)O
World Health Organisation international non-proprietary name
olodaterol
subject has role
bronchodilator
defined daily dose
5.0
physically interacts with
adrenoceptor beta 2
Commons category
Olodaterol
Sources (3)

via Wikidata · CC0

~6 min read

Encyclopedic overview

10 sections
Contents
  • Medical uses
  • Adverse effects
  • Interactions
  • Pharmacology
  • Mechanism of action
  • Pharmacokinetics
  • Pharmacodynamics
  • History
  • References
  • External links

{{Drugbox | IUPAC_name = 6-hydroxy-8-{(1R)-1-hydroxy-2-{[1-(4-methoxyphenyl)-2-methylpropan-2-yl]amino}ethyl}-4H-1,4-benzoxazin-3-one | image = Olodaterol skeletal.svg | image_class = skin-invert-image | width = 275 | alt = | caption = | tradename = Striverdi Respimat | pronounce = Striverdi Respimat | Drugs.com = | MedlinePlus = | pregnancy_AU = B3 | pregnancy_US = C | legal_AU = S4 | legal_CA = | legal_UK = POM | legal_US = Rx-only | legal_status = Rx-only | routes_of_administration = Inhalation (MDI)

| bioavailability = ~30% (inhalation) | protein_bound = ~60% | metabolism = Liver | elimination_half-life = 7.5 hours | excretion = Feces (53%), urine (38%) — following IV administration

Excerpted from Wikipedia’s “olodaterol” article, available under the CC BY-SA 4.0 licence.