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EntityQ2602750· pop 19· linked from 507 articles

diflunisal

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Also known as 5-(2,4-difluorophenyl)salicylic acid, 2-(hydroxy)-5-(2,4-difluorophenyl)benzoic acid, 2',4'-difluoro-4-hydroxy-3-biphenylcarboxylic acid

Diflunisal is a salicylic acid derivative with analgesic and anti-inflammatory activity. It was developed by Merck Sharp & Dohme in 1971, after showing promise in a research project studying more potent chemical analogs of aspirin. It was first sold under the brand name Dolobid, by Merck & Co., but generic versions are widely available. It is classed as a nonsteroidal anti-inflammatory drug (NSAID) and is available in 250 mg and 500 mg tablets.

Key facts

Drug.verifiedrevid
460785966
Drug.image
Diflunisal structure.svg
Drug.width
180
Drug.image_class
skin-invert-image
Drug.image2
Diflunasil-3D-balls.png
Drug.width2
187
Drug.image_class2
bg-transparent
Drug.tradename
Dolobid
Drug.MedlinePlus
a684037
Drug.DailyMedID
Diflunisal
Drug.pregnancy_AU
C
Drug.routes_of_administration
By mouth
Drug.ATC_prefix
N02
Drug.ATC_suffix
BA11
Drug.legal_AU
S4
Drug.legal_UK
POM
Drug.legal_US
Rx-only
Drug.legal_EU
Rx-only

via Wikipedia infobox

Wikidata facts

Mass
250.044
Has use
medication
Show 8 more facts
World Health Organisation international non-proprietary name
diflunisal
chemical formula
C₁₃H₈F₂O₃
medical condition treated
rheumatoid arthritis
canonical SMILES
C1=CC(=C(C=C1C2=C(C=C(C=C2)F)F)C(=O)O)O
defined daily dose
0.75
Commons category
Diflunisal
physically interacts with
Prostaglandin-endoperoxide synthase 1
legal status (medicine)
boxed warning
Sources (8)

via Wikidata · CC0

~3 min read

Encyclopedic overview

11 sections
Contents
  • Medical uses
  • Contraindications
  • Amyloidosis
  • Side effects
  • Mechanism of action
  • Duration of effect
  • Society and culture
  • Legal status
  • Research
  • References
  • Further reading

Diflunisal is a salicylic acid derivative with analgesic and anti-inflammatory activity. It was developed by Merck Sharp & Dohme in 1971, after showing promise in a research project studying more potent chemical analogs of aspirin. It was first sold under the brand name Dolobid, by Merck & Co., but generic versions are widely available. It is classed as a nonsteroidal anti-inflammatory drug (NSAID) and is available in 250 mg and 500 mg tablets.

==Medical uses== Diflunisal is indicated for acute or long-term use for symptomatic treatment of mild to moderate pain, osteoarthritis, and rheumatoid arthritis.

Excerpted from Wikipedia’s “diflunisal” article, available under the CC BY-SA 4.0 licence.