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tolpiprazole

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tolpiprazole

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Tolpiprazole (INN, BAN) (developmental code name H-4170) is an anxiolytic drug of the phenylpiperazine group that was never marketed.

Chemical data

Formula
C17H24N4
Molecular weight
284.4 g/mol
IUPAC name
1-(3-methylphenyl)-4-[2-(5-methyl-1H-pyrazol-3-yl)ethyl]piperazine
SMILES
CC1=CC(=CC=C1)N2CCN(CC2)CCC3=NNC(=C3)C
InChIKey
IYBFBADVQPQHLQ-UHFFFAOYSA-N
XLogP
2.9
Polar surface area
35.2 Ų
H-bond donors
1
H-bond acceptors
3
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Phase 2
Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
284.2
Show 2 more facts
chemical formula
C₁₇H₂₄N₄
canonical SMILES
CC1=CC(=CC=C1)N2CCN(CC2)CCC3=NNC(=C3)C
Sources (2)

via Wikidata · CC0

~1 min read

Encyclopedic overview

2 sections
Contents
  • See also
  • References

Tolpiprazole (INN, BAN) (developmental code name H-4170) is an anxiolytic drug of the phenylpiperazine group that was never marketed.

==See also== Acaprazine Enpiprazole Lorpiprazole Mepiprazole

Excerpted from Wikipedia’s “tolpiprazole” article, available under the CC BY-SA 4.0 licence.

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