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erdosteine

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Erdosteine is a molecule with mucolytic activity. Structurally it is a thioether derivative with two thioether groups. These two functional organosulfur groups contained in the molecule are released following first-pass metabolism with the conversion of erdosteine into its pharmacologically active metabolite Met-I (N-thiodiglycolyl-homocysteine).

Wikidata facts

Mass
249.013
Show 3 more facts
chemical formula
C₈H₁₁NO₄S₂
canonical SMILES
C1CSC(=O)C1NC(=O)CSCC(=O)O
Commons category
Erdosteine
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Article

14 sections
Contents
  • Pharmacodynamics
  • [[Antioxidant|Anti-oxidant]] and [[anti-inflammatory]] activity
  • Antiadhesive activity
  • [[Mucoactive agent|Mucolytic]] activity
  • [[Chronic obstructive pulmonary disease|Chronic Obstructive Pulmonary Disease]]
  • Other activities
  • Pediatric population
  • Pharmacokinetics
  • Toxicity
  • Clinical uses
  • Safety profile
  • Contraindications
  • Interaction with other medicinal products
  • References

Erdosteine is a molecule with mucolytic activity. Structurally it is a thioether derivative with two thioether groups. These two functional organosulfur groups contained in the molecule are released following first-pass metabolism with the conversion of erdosteine into its pharmacologically active metabolite Met-I (N-thiodiglycolyl-homocysteine).

The molecule has been discovered and developed in Italy by Edmond Pharma, today it is prescribed for chronic and acute respiratory disorders in more than 40 countries worldwide. The drug is sold under several commercial names (Esteclin, Erdomed, Erdos, Erdotin etc.), as hard capsules 300 mg, dispersible tablets 300 mg, granulates for oral suspension 225 mg and powder for oral suspension 175 mg/5ml.

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