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nitecapone

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nitecapone

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Nitecapone (INN; OR-462) is a drug which acts as a selective inhibitor of the enzyme catechol O-methyl transferase (COMT). It was patented as an antiparkinson medication but was never marketed.

Chemical data

Formula
C12H11NO6
Molecular weight
265.22 g/mol
IUPAC name
3-[(3,4-dihydroxy-5-nitrophenyl)methylidene]pentane-2,4-dione
SMILES
CC(=O)C(=CC1=CC(=C(C(=C1)O)O)[N+](=O)[O-])C(=O)C
InChIKey
UPMRZALMHVUCIN-UHFFFAOYSA-N
XLogP
1.2
Polar surface area
120 Ų
H-bond donors
2
H-bond acceptors
6
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Phase 2
Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
265.059
Has use
medication
Show 4 more facts
chemical formula
C₁₂H₁₁NO₆
canonical SMILES
CC(=O)C(=CC1=CC(=C(C(=C1)O)O)[N+](=O)[O-])C(=O)C
subject has role
antioxidant
Commons category
Nitecapone
Sources (2)

via Wikidata · CC0

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Encyclopedic overview

2 sections
Contents
  • See also
  • References

Nitecapone (INN; OR-462) is a drug which acts as a selective inhibitor of the enzyme catechol O-methyl transferase (COMT). It was patented as an antiparkinson medication but was never marketed.

==See also== List of investigational Parkinson's disease drugs Catechol-O-methyltransferase inhibitor

Excerpted from Wikipedia’s “nitecapone” article, available under the CC BY-SA 4.0 licence.

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