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paliperidone

Structure via PubChem · Public domain (PubChem)

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paliperidone

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Also known as 9-hydroxyrisperidone, Invega®, Ro-76477, Ro-92670, Trevicta, 9-Hydroxyrisperidone

Paliperidone, sold under the brand name Invega among others, is an atypical antipsychotic. It is used for the treatment of schizophrenia and schizoaffective disorder. It is marketed by Janssen Pharmaceuticals.

Key facts

Drug.Verifiedfields
changed
Drug.Watchedfields
changed
Drug.verifiedrevid
461753832
Drug.image
Paliperidone.svg
Drug.image_class
skin-invert-image
Drug.width
250
Drug.tradename
Invega, others
Drug.MedlinePlus
a607005
Drug.DailyMedID
Paliperidone
Drug.pregnancy_AU
B3
Drug.routes_of_administration
By mouth, intramuscular
Drug.class
Atypical antipsychotic
Drug.ATC_prefix
N05
Drug.ATC_suffix
AX13
Drug.legal_AU
S4
Drug.legal_BR
C1
Drug.legal_CA
Rx-only
Drug.legal_US
Rx-only

via Wikipedia infobox

Chemical data

Formula
C23H27FN4O3
Molecular weight
426.5 g/mol
IUPAC name
3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-9-hydroxy-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one
SMILES
CC1=C(C(=O)N2CCCC(C2=N1)O)CCN3CCC(CC3)C4=NOC5=C4C=CC(=C5)F
InChIKey
PMXMIIMHBWHSKN-UHFFFAOYSA-N
XLogP
2.2
Polar surface area
82.2 Ų
H-bond donors
1
H-bond acceptors
7
Formal charge
0

via PubChem

Wikidata facts

Mass
426.206719
Show 4 more facts
chemical formula
C₂₃H₂₇FN₄O₃
Commons category
Paliperidone
canonical SMILES
CC1=C(C(=O)N2CCCC(C2=N1)O)CCN3CCC(CC3)C4=NOC5=C4C=CC(=C5)F
defined daily dose
2.5
Sources (6)

via Wikidata · CC0

~7 min read

Article

11 sections
Contents
  • Medical use
  • Adverse effects
  • Pharmacology
  • History
  • Society and culture
  • Deaths
  • Suicides
  • Homicides
  • Brand names
  • References
  • External links

Paliperidone, sold under the brand name Invega among others, is an atypical antipsychotic. It is used for the treatment of schizophrenia and schizoaffective disorder. It is marketed by Janssen Pharmaceuticals.

Paliperidone was approved by the US Food and Drug Administration (FDA) for the treatment of schizophrenia in December 2006, and in the European Union in June 2007. Paliperidone palmitate is a long-acting injectable formulation of paliperidone palmitoyl ester. It is on the World Health Organization's List of Essential Medicines. Paliperidone is available as a generic medication.

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